Ring-opened tetrahydro-γ-carbolines display cytotoxicity and selectivity with histone deacetylase isoforms.

Nepali, Kunal

Ring-opened tetrahydro-γ-carbolines display cytotoxicity and selectivity with histone deacetylase isoforms. [electronic resource] - European journal of medicinal chemistry Feb 2017 - 115-127 p. digital

Publication Type: Journal Article

1768-3254

10.1016/j.ejmech.2016.12.039 doi


Antineoplastic Agents--chemistry
Apoptosis--drug effects
Carbolines--chemistry
Cell Line, Tumor
Cell Proliferation--drug effects
Histone Deacetylase Inhibitors--chemistry
Histone Deacetylases--metabolism
Humans
Isoenzymes--antagonists & inhibitors
Structure-Activity Relationship