Synthesis and biological evaluation of N-(3-oxo-3,4-dihydro-2H-benzo[b][1,4]oxazin-7-yl)benzenesulfonamide derivatives as new BET bromodomain inhibitors for anti-hematologic malignancies activities.

Liu, Li

Synthesis and biological evaluation of N-(3-oxo-3,4-dihydro-2H-benzo[b][1,4]oxazin-7-yl)benzenesulfonamide derivatives as new BET bromodomain inhibitors for anti-hematologic malignancies activities. [electronic resource] - Molecular diversity Feb 2017 - 125-136 p. digital

Publication Type: Journal Article

1573-501X

10.1007/s11030-016-9707-6 doi


Antineoplastic Agents--chemical synthesis
Cell Line, Tumor
Epigenesis, Genetic
Hematologic Neoplasms--pathology
Humans
Protein Domains
Structure-Activity Relationship
Sulfonamides--chemical synthesis
Benzenesulfonamides