A TPX2 Proteomimetic Has Enhanced Affinity for Aurora-A Due to Hydrocarbon Stapling of a Helix.

Rennie, Yana K

A TPX2 Proteomimetic Has Enhanced Affinity for Aurora-A Due to Hydrocarbon Stapling of a Helix. [electronic resource] - ACS chemical biology 12 2016 - 3383-3390 p. digital

Publication Type: Journal Article; Research Support, Non-U.S. Gov't

1554-8937

10.1021/acschembio.6b00727 doi


Amino Acid Sequence
Aurora Kinase A--chemistry
Cell Cycle Proteins--chemistry
Crystallography, X-Ray
Enzyme Activation
Humans
Microtubule-Associated Proteins--chemistry
Molecular Docking Simulation
Nuclear Proteins--chemistry
Protein Binding
Protein Conformation, alpha-Helical
Protein Interaction Maps
Thermodynamics