The Dual Syk/JAK Inhibitor Cerdulatinib Antagonizes B-cell Receptor and Microenvironmental Signaling in Chronic Lymphocytic Leukemia.
Blunt, Matthew D
The Dual Syk/JAK Inhibitor Cerdulatinib Antagonizes B-cell Receptor and Microenvironmental Signaling in Chronic Lymphocytic Leukemia. [electronic resource] - Clinical cancer research : an official journal of the American Association for Cancer Research May 2017 - 2313-2324 p. digital
Publication Type: Journal Article
1557-3265
10.1158/1078-0432.CCR-16-1662 doi
Adenine--analogs & derivatives
Antineoplastic Combined Chemotherapy Protocols--administration & dosage
Apoptosis--drug effects
B-Lymphocytes--drug effects
Bridged Bicyclo Compounds, Heterocyclic--administration & dosage
Flow Cytometry
Gene Expression Regulation, Neoplastic--drug effects
Humans
Janus Kinase Inhibitors--administration & dosage
Janus Kinases--antagonists & inhibitors
Leukemia, Lymphocytic, Chronic, B-Cell--drug therapy
Leukocytes, Mononuclear--drug effects
Neoplasm Proteins--genetics
Piperidines
Proto-Oncogene Proteins c-bcr--antagonists & inhibitors
Pyrazoles--administration & dosage
Pyrimidines--administration & dosage
Receptors, Antigen, B-Cell--drug effects
Signal Transduction--drug effects
Sulfonamides--administration & dosage
Sulfones--administration & dosage
Syk Kinase--antagonists & inhibitors
Tumor Microenvironment--drug effects
The Dual Syk/JAK Inhibitor Cerdulatinib Antagonizes B-cell Receptor and Microenvironmental Signaling in Chronic Lymphocytic Leukemia. [electronic resource] - Clinical cancer research : an official journal of the American Association for Cancer Research May 2017 - 2313-2324 p. digital
Publication Type: Journal Article
1557-3265
10.1158/1078-0432.CCR-16-1662 doi
Adenine--analogs & derivatives
Antineoplastic Combined Chemotherapy Protocols--administration & dosage
Apoptosis--drug effects
B-Lymphocytes--drug effects
Bridged Bicyclo Compounds, Heterocyclic--administration & dosage
Flow Cytometry
Gene Expression Regulation, Neoplastic--drug effects
Humans
Janus Kinase Inhibitors--administration & dosage
Janus Kinases--antagonists & inhibitors
Leukemia, Lymphocytic, Chronic, B-Cell--drug therapy
Leukocytes, Mononuclear--drug effects
Neoplasm Proteins--genetics
Piperidines
Proto-Oncogene Proteins c-bcr--antagonists & inhibitors
Pyrazoles--administration & dosage
Pyrimidines--administration & dosage
Receptors, Antigen, B-Cell--drug effects
Signal Transduction--drug effects
Sulfonamides--administration & dosage
Sulfones--administration & dosage
Syk Kinase--antagonists & inhibitors
Tumor Microenvironment--drug effects