Oncogenic Receptor Tyrosine Kinases Directly Phosphorylate Focal Adhesion Kinase (FAK) as a Resistance Mechanism to FAK-Kinase Inhibitors.

Marlowe, Timothy A

Oncogenic Receptor Tyrosine Kinases Directly Phosphorylate Focal Adhesion Kinase (FAK) as a Resistance Mechanism to FAK-Kinase Inhibitors. [electronic resource] - Molecular cancer therapeutics 12 2016 - 3028-3039 p. digital

Publication Type: Journal Article

1538-8514

10.1158/1535-7163.MCT-16-0366 doi


Antineoplastic Agents--chemistry
Cell Line, Tumor
Cell Movement--genetics
Drug Resistance, Neoplasm
ErbB Receptors--chemistry
Focal Adhesion Protein-Tyrosine Kinases--antagonists & inhibitors
Gene Knockout Techniques
Humans
Phosphorylation
Protein Binding
Protein Kinase Inhibitors--chemistry
Receptor Protein-Tyrosine Kinases--chemistry
Receptor, ErbB-2--chemistry
Signal Transduction--drug effects