Identification and Optimization of the First Highly Selective GLUT1 Inhibitor BAY-876.

Siebeneicher, Holger

Identification and Optimization of the First Highly Selective GLUT1 Inhibitor BAY-876. [electronic resource] - ChemMedChem 10 2016 - 2261-2271 p. digital

Publication Type: Journal Article

1860-7187

10.1002/cmdc.201600276 doi


Administration, Oral
Biological Availability
Glucose Transporter Type 1--antagonists & inhibitors
High-Throughput Screening Assays
Humans
Molecular Structure
Pyrazoles--administration & dosage
Quinolines--administration & dosage
Structure-Activity Relationship