Discovery, characterization, and lead optimization of 7-azaindole non-nucleoside HIV-1 reverse transcriptase inhibitors.

Stanton, Richard A

Discovery, characterization, and lead optimization of 7-azaindole non-nucleoside HIV-1 reverse transcriptase inhibitors. [electronic resource] - Bioorganic & medicinal chemistry letters 08 2016 - 4101-5 p. digital

Publication Type: Journal Article

1464-3405

10.1016/j.bmcl.2016.06.065 doi


Animals
Binding Sites
Cell Survival--drug effects
Chlorocebus aethiops
Drug Evaluation, Preclinical
HIV Reverse Transcriptase--antagonists & inhibitors
HIV-1--drug effects
Humans
Indoles--chemistry
Molecular Docking Simulation
Mutagenesis, Site-Directed
Protein Binding
Protein Structure, Tertiary
Reverse Transcriptase Inhibitors--chemistry
Vero Cells