DNA sequence-selective C8-linked pyrrolobenzodiazepine-heterocyclic polyamide conjugates show anti-tubercular-specific activities.

Brucoli, Federico

DNA sequence-selective C8-linked pyrrolobenzodiazepine-heterocyclic polyamide conjugates show anti-tubercular-specific activities. [electronic resource] - The Journal of antibiotics Dec 2016 - 843-849 p. digital

Publication Type: Journal Article

1881-1469

10.1038/ja.2016.43 doi


Animals
Antitubercular Agents--pharmacology
Base Sequence
Benzodiazepines--chemistry
DNA Footprinting
DNA, Bacterial--genetics
Deoxyribonuclease I--genetics
Escherichia coli--drug effects
Isoniazid--pharmacology
Mice
Microbial Sensitivity Tests
Mycobacterium bovis--drug effects
Mycobacterium tuberculosis--drug effects
Nylons--chemistry
Pseudomonas putida--drug effects
Pyrroles--chemistry
RAW 264.7 Cells
Rhodococcus--drug effects
Rifampin--pharmacology
Sequence Analysis, DNA