Bioavailable inhibitors of HIV-1 RNA biogenesis identified through a Rev-based screen.
Prado, Silvia
Bioavailable inhibitors of HIV-1 RNA biogenesis identified through a Rev-based screen. [electronic resource] - Biochemical pharmacology May 2016 - 14-28 p. digital
Publication Type: Journal Article; Research Support, Non-U.S. Gov't
1873-2968
10.1016/j.bcp.2016.02.007 doi
Anti-HIV Agents--adverse effects
Cell Line
Cell Survival--drug effects
Clomiphene--adverse effects
Cyproheptadine--adverse effects
Drug Evaluation, Preclinical
Gene Expression Regulation, Viral--drug effects
Genes, Reporter--drug effects
HIV-1--drug effects
High-Throughput Screening Assays
Humans
Peptide Fragments--antagonists & inhibitors
Protein Interaction Domains and Motifs
RNA Splicing--drug effects
RNA, Viral--metabolism
Recombinant Proteins--chemistry
Response Elements--drug effects
Small Molecule Libraries
Transcription, Genetic--drug effects
rev Gene Products, Human Immunodeficiency Virus--antagonists & inhibitors
Bioavailable inhibitors of HIV-1 RNA biogenesis identified through a Rev-based screen. [electronic resource] - Biochemical pharmacology May 2016 - 14-28 p. digital
Publication Type: Journal Article; Research Support, Non-U.S. Gov't
1873-2968
10.1016/j.bcp.2016.02.007 doi
Anti-HIV Agents--adverse effects
Cell Line
Cell Survival--drug effects
Clomiphene--adverse effects
Cyproheptadine--adverse effects
Drug Evaluation, Preclinical
Gene Expression Regulation, Viral--drug effects
Genes, Reporter--drug effects
HIV-1--drug effects
High-Throughput Screening Assays
Humans
Peptide Fragments--antagonists & inhibitors
Protein Interaction Domains and Motifs
RNA Splicing--drug effects
RNA, Viral--metabolism
Recombinant Proteins--chemistry
Response Elements--drug effects
Small Molecule Libraries
Transcription, Genetic--drug effects
rev Gene Products, Human Immunodeficiency Virus--antagonists & inhibitors