Tricyclic pyrazoles. Part 8. Synthesis, biological evaluation and modelling of tricyclic pyrazole carboxamides as potential CB2 receptor ligands with antagonist/inverse agonist properties.

Deiana, Valeria

Tricyclic pyrazoles. Part 8. Synthesis, biological evaluation and modelling of tricyclic pyrazole carboxamides as potential CB2 receptor ligands with antagonist/inverse agonist properties. [electronic resource] - European journal of medicinal chemistry Apr 2016 - 66-80 p. digital

Publication Type: Journal Article; Research Support, Non-U.S. Gov't

1768-3254

10.1016/j.ejmech.2016.02.005 doi


Humans
Ligands
Molecular Docking Simulation
Pyrazoles--chemical synthesis
Receptor, Cannabinoid, CB2--agonists
Structure-Activity Relationship