Design and optimization of tricyclic gamma-secretase modulators.

Shi, Jianliang

Design and optimization of tricyclic gamma-secretase modulators. [electronic resource] - Bioorganic & medicinal chemistry letters Mar 2016 - 1498-502 p. digital

Publication Type: Journal Article

1464-3405

10.1016/j.bmcl.2015.06.020 doi


Amyloid Precursor Protein Secretases--antagonists & inhibitors
Aniline Compounds--chemical synthesis
Animals
Dose-Response Relationship, Drug
Drug Design
Humans
Mice
Molecular Structure
Protease Inhibitors--chemical synthesis
Structure-Activity Relationship
Triazines--chemical synthesis