Optimisation of a triazolopyridine based histone demethylase inhibitor yields a potent and selective KDM2A (FBXL11) inhibitor.

England, Katherine S

Optimisation of a triazolopyridine based histone demethylase inhibitor yields a potent and selective KDM2A (FBXL11) inhibitor. [electronic resource] - MedChemComm Dec 2014 - 1879-1886 p. digital

Publication Type: Journal Article

2040-2503

10.1039/C4MD00291A doi