Transcriptional Profiling of a Selective CREB Binding Protein Bromodomain Inhibitor Highlights Therapeutic Opportunities.
Chekler, Eugene L Piatnitski
Transcriptional Profiling of a Selective CREB Binding Protein Bromodomain Inhibitor Highlights Therapeutic Opportunities. [electronic resource] - Chemistry & biology Dec 2015 - 1588-96 p. digital
Publication Type: Journal Article
1879-1301
10.1016/j.chembiol.2015.10.013 doi
CREB-Binding Protein--antagonists & inhibitors
Drug Design
Fluorescence Resonance Energy Transfer
Gene Expression Regulation--drug effects
Humans
Protein Structure, Tertiary
RGS Proteins--genetics
Small Molecule Libraries--chemistry
Transcriptome
Transcriptional Profiling of a Selective CREB Binding Protein Bromodomain Inhibitor Highlights Therapeutic Opportunities. [electronic resource] - Chemistry & biology Dec 2015 - 1588-96 p. digital
Publication Type: Journal Article
1879-1301
10.1016/j.chembiol.2015.10.013 doi
CREB-Binding Protein--antagonists & inhibitors
Drug Design
Fluorescence Resonance Energy Transfer
Gene Expression Regulation--drug effects
Humans
Protein Structure, Tertiary
RGS Proteins--genetics
Small Molecule Libraries--chemistry
Transcriptome