Development of Bifunctional Inhibitors of Polo-Like Kinase 1 with Low-Nanomolar Activities Against the Polo-Box Domain.
Scharow, Andrej
Development of Bifunctional Inhibitors of Polo-Like Kinase 1 with Low-Nanomolar Activities Against the Polo-Box Domain. [electronic resource] - Chembiochem : a European journal of chemical biology Apr 2016 - 759-67 p. digital
Publication Type: Journal Article; Research Support, Non-U.S. Gov't
1439-7633
10.1002/cbic.201500535 doi
Cell Cycle Proteins--antagonists & inhibitors
Dose-Response Relationship, Drug
Fluorescence Polarization
Humans
Molecular Structure
Peptides--chemical synthesis
Protein Kinase Inhibitors--chemistry
Protein Serine-Threonine Kinases--antagonists & inhibitors
Proto-Oncogene Proteins--antagonists & inhibitors
Structure-Activity Relationship
Polo-Like Kinase 1
Development of Bifunctional Inhibitors of Polo-Like Kinase 1 with Low-Nanomolar Activities Against the Polo-Box Domain. [electronic resource] - Chembiochem : a European journal of chemical biology Apr 2016 - 759-67 p. digital
Publication Type: Journal Article; Research Support, Non-U.S. Gov't
1439-7633
10.1002/cbic.201500535 doi
Cell Cycle Proteins--antagonists & inhibitors
Dose-Response Relationship, Drug
Fluorescence Polarization
Humans
Molecular Structure
Peptides--chemical synthesis
Protein Kinase Inhibitors--chemistry
Protein Serine-Threonine Kinases--antagonists & inhibitors
Proto-Oncogene Proteins--antagonists & inhibitors
Structure-Activity Relationship
Polo-Like Kinase 1