Development of Potent and Selective Tissue Transglutaminase Inhibitors: Their Effect on TG2 Function and Application in Pathological Conditions.

Badarau, Eduard

Development of Potent and Selective Tissue Transglutaminase Inhibitors: Their Effect on TG2 Function and Application in Pathological Conditions. [electronic resource] - Chemistry & biology Oct 2015 - 1347-61 p. digital

Publication Type: Journal Article; Research Support, Non-U.S. Gov't

1879-1301

10.1016/j.chembiol.2015.08.013 doi


Animals
Blotting, Western
Endothelial Cells--drug effects
Enzyme Activation--drug effects
Enzyme Inhibitors--chemistry
Fibrosis--drug therapy
GTP-Binding Proteins--antagonists & inhibitors
Humans
Mice
Mice, Inbred C57BL
Microscopy, Fluorescence
NIH 3T3 Cells
Nephrosclerosis--drug therapy
Protein Binding--drug effects
Protein Glutamine gamma Glutamyltransferase 2
Small Molecule Libraries--chemistry
Syndecan-4--metabolism
Transglutaminases--antagonists & inhibitors