6-Methyluracil Derivatives as Bifunctional Acetylcholinesterase Inhibitors for the Treatment of Alzheimer's Disease.

Semenov, Vyacheslav E

6-Methyluracil Derivatives as Bifunctional Acetylcholinesterase Inhibitors for the Treatment of Alzheimer's Disease. [electronic resource] - ChemMedChem Nov 2015 - 1863-74 p. digital

Publication Type: Journal Article; Research Support, Non-U.S. Gov't

1860-7187

10.1002/cmdc.201500334 doi


Acetylcholinesterase--metabolism
Alzheimer Disease--drug therapy
Animals
Behavior, Animal--drug effects
Brain--enzymology
Cholinesterase Inhibitors--chemical synthesis
Crystallography, X-Ray
Disease Models, Animal
Dose-Response Relationship, Drug
Humans
Mice
Mice, Transgenic
Models, Molecular
Molecular Structure
Structure-Activity Relationship
Uracil--analogs & derivatives