Selective Targeting of Extracellular Insulin-Degrading Enzyme by Quasi-Irreversible Thiol-Modifying Inhibitors.
Abdul-Hay, Samer O
Selective Targeting of Extracellular Insulin-Degrading Enzyme by Quasi-Irreversible Thiol-Modifying Inhibitors. [electronic resource] - ACS chemical biology Dec 2015 - 2716-24 p. digital
Publication Type: Journal Article
1554-8937
10.1021/acschembio.5b00334 doi
Computer Simulation
Cytosol--chemistry
Drug Delivery Systems
Drug Evaluation, Preclinical
Enzyme Inhibitors--chemical synthesis
Extracellular Space--enzymology
Inhibitory Concentration 50
Insulin Antagonists--pharmacology
Insulysin--antagonists & inhibitors
Models, Biological
Molecular Structure
Structure-Activity Relationship
Sulfhydryl Compounds--chemistry
Selective Targeting of Extracellular Insulin-Degrading Enzyme by Quasi-Irreversible Thiol-Modifying Inhibitors. [electronic resource] - ACS chemical biology Dec 2015 - 2716-24 p. digital
Publication Type: Journal Article
1554-8937
10.1021/acschembio.5b00334 doi
Computer Simulation
Cytosol--chemistry
Drug Delivery Systems
Drug Evaluation, Preclinical
Enzyme Inhibitors--chemical synthesis
Extracellular Space--enzymology
Inhibitory Concentration 50
Insulin Antagonists--pharmacology
Insulysin--antagonists & inhibitors
Models, Biological
Molecular Structure
Structure-Activity Relationship
Sulfhydryl Compounds--chemistry