2,4-Diarylamino-pyrimidines as kinase inhibitors co-targeting IGF1R and EGFR(L⁸⁵⁸R/T⁷⁹⁰M).
Chan, Shingpan
2,4-Diarylamino-pyrimidines as kinase inhibitors co-targeting IGF1R and EGFR(L⁸⁵⁸R/T⁷⁹⁰M). [electronic resource] - Bioorganic & medicinal chemistry letters Oct 2015 - 4277-81 p. digital
Publication Type: Journal Article; Research Support, Non-U.S. Gov't
1464-3405
10.1016/j.bmcl.2015.07.089 doi
Antineoplastic Agents--chemical synthesis
Cell Line, Tumor
Cell Proliferation--drug effects
Dose-Response Relationship, Drug
Drug Screening Assays, Antitumor
ErbB Receptors--antagonists & inhibitors
Humans
Models, Molecular
Molecular Structure
Protein Kinase Inhibitors--chemical synthesis
Receptor, IGF Type 1
Receptors, Somatomedin--antagonists & inhibitors
Structure-Activity Relationship
2,4-Diarylamino-pyrimidines as kinase inhibitors co-targeting IGF1R and EGFR(L⁸⁵⁸R/T⁷⁹⁰M). [electronic resource] - Bioorganic & medicinal chemistry letters Oct 2015 - 4277-81 p. digital
Publication Type: Journal Article; Research Support, Non-U.S. Gov't
1464-3405
10.1016/j.bmcl.2015.07.089 doi
Antineoplastic Agents--chemical synthesis
Cell Line, Tumor
Cell Proliferation--drug effects
Dose-Response Relationship, Drug
Drug Screening Assays, Antitumor
ErbB Receptors--antagonists & inhibitors
Humans
Models, Molecular
Molecular Structure
Protein Kinase Inhibitors--chemical synthesis
Receptor, IGF Type 1
Receptors, Somatomedin--antagonists & inhibitors
Structure-Activity Relationship