Identification of orally-bioavailable antagonists of the TRPV4 ion-channel.
Wei, Zhi-Liang
Identification of orally-bioavailable antagonists of the TRPV4 ion-channel. [electronic resource] - Bioorganic & medicinal chemistry letters Sep 2015 - 4011-5 p. digital
Publication Type: Journal Article
1464-3405
10.1016/j.bmcl.2015.06.098 doi
Administration, Oral
Animals
Biological Availability
Dose-Response Relationship, Drug
Humans
Mice
Molecular Structure
Piperazines--administration & dosage
Rats
Rats, Wistar
Structure-Activity Relationship
TRPV Cation Channels--antagonists & inhibitors
Identification of orally-bioavailable antagonists of the TRPV4 ion-channel. [electronic resource] - Bioorganic & medicinal chemistry letters Sep 2015 - 4011-5 p. digital
Publication Type: Journal Article
1464-3405
10.1016/j.bmcl.2015.06.098 doi
Administration, Oral
Animals
Biological Availability
Dose-Response Relationship, Drug
Humans
Mice
Molecular Structure
Piperazines--administration & dosage
Rats
Rats, Wistar
Structure-Activity Relationship
TRPV Cation Channels--antagonists & inhibitors