Identification of orally-bioavailable antagonists of the TRPV4 ion-channel.

Wei, Zhi-Liang

Identification of orally-bioavailable antagonists of the TRPV4 ion-channel. [electronic resource] - Bioorganic & medicinal chemistry letters Sep 2015 - 4011-5 p. digital

Publication Type: Journal Article

1464-3405

10.1016/j.bmcl.2015.06.098 doi


Administration, Oral
Animals
Biological Availability
Dose-Response Relationship, Drug
Humans
Mice
Molecular Structure
Piperazines--administration & dosage
Rats
Rats, Wistar
Structure-Activity Relationship
TRPV Cation Channels--antagonists & inhibitors