Identification of a DYRK1A Inhibitor that Induces Degradation of the Target Kinase using Co-chaperone CDC37 fused with Luciferase nanoKAZ.
Sonamoto, Rie
Identification of a DYRK1A Inhibitor that Induces Degradation of the Target Kinase using Co-chaperone CDC37 fused with Luciferase nanoKAZ. [electronic resource] - Scientific reports Aug 2015 - 12728 p. digital
Publication Type: Journal Article; Research Support, Non-U.S. Gov't
2045-2322
10.1038/srep12728 doi
Benzofurans--pharmacology
Cell Cycle Proteins--genetics
Chaperonins--genetics
Drug Evaluation, Preclinical--methods
HEK293 Cells
HSP90 Heat-Shock Proteins--genetics
Humans
Luciferases--genetics
Molecular Chaperones--genetics
Mutation
Protein Kinase Inhibitors--pharmacology
Protein Serine-Threonine Kinases--antagonists & inhibitors
Protein-Tyrosine Kinases--antagonists & inhibitors
Recombinant Fusion Proteins--genetics
Small Molecule Libraries--pharmacology
Thiazolidines--pharmacology
Triazoles--pharmacology
Dyrk Kinases
Identification of a DYRK1A Inhibitor that Induces Degradation of the Target Kinase using Co-chaperone CDC37 fused with Luciferase nanoKAZ. [electronic resource] - Scientific reports Aug 2015 - 12728 p. digital
Publication Type: Journal Article; Research Support, Non-U.S. Gov't
2045-2322
10.1038/srep12728 doi
Benzofurans--pharmacology
Cell Cycle Proteins--genetics
Chaperonins--genetics
Drug Evaluation, Preclinical--methods
HEK293 Cells
HSP90 Heat-Shock Proteins--genetics
Humans
Luciferases--genetics
Molecular Chaperones--genetics
Mutation
Protein Kinase Inhibitors--pharmacology
Protein Serine-Threonine Kinases--antagonists & inhibitors
Protein-Tyrosine Kinases--antagonists & inhibitors
Recombinant Fusion Proteins--genetics
Small Molecule Libraries--pharmacology
Thiazolidines--pharmacology
Triazoles--pharmacology
Dyrk Kinases