Human hepatocyte assessment of imatinib drug-drug interactions - complexities in clinical translation.

Beumer, Jan H

Human hepatocyte assessment of imatinib drug-drug interactions - complexities in clinical translation. [electronic resource] - British journal of clinical pharmacology Nov 2015 - 1097-108 p. digital

Publication Type: Journal Article; Research Support, N.I.H., Extramural

1365-2125

10.1111/bcp.12723 doi


Adolescent
Adult
Aged
Alkynes
Anti-HIV Agents--pharmacology
Benzoxazines--pharmacology
Cyclopropanes
Cytochrome P-450 CYP3A Inducers--pharmacology
Cytochrome P-450 CYP3A Inhibitors--pharmacology
Drug Interactions
Female
Hepatocytes--cytology
Humans
Imatinib Mesylate--metabolism
Ketoconazole--pharmacology
Male
Middle Aged
Primary Cell Culture
Rifampin--pharmacology
Ritonavir--pharmacology
Young Adult