Design, synthesis and biological evaluation of small molecules as potent glucosidase inhibitors.
Hati, Santanu
Design, synthesis and biological evaluation of small molecules as potent glucosidase inhibitors. [electronic resource] - European journal of medicinal chemistry Jul 2015 - 188-96 p. digital
Publication Type: Journal Article; Research Support, Non-U.S. Gov't
1768-3254
10.1016/j.ejmech.2015.04.059 doi
Antimalarials--chemical synthesis
Dose-Response Relationship, Drug
Drug Design
Enzyme Inhibitors--chemical synthesis
Glucosidases--antagonists & inhibitors
Humans
Malaria, Falciparum--drug therapy
Models, Molecular
Molecular Structure
Parasitic Sensitivity Tests
Plasmodium falciparum--drug effects
Saccharomyces cerevisiae--enzymology
Small Molecule Libraries--chemical synthesis
Structure-Activity Relationship
Design, synthesis and biological evaluation of small molecules as potent glucosidase inhibitors. [electronic resource] - European journal of medicinal chemistry Jul 2015 - 188-96 p. digital
Publication Type: Journal Article; Research Support, Non-U.S. Gov't
1768-3254
10.1016/j.ejmech.2015.04.059 doi
Antimalarials--chemical synthesis
Dose-Response Relationship, Drug
Drug Design
Enzyme Inhibitors--chemical synthesis
Glucosidases--antagonists & inhibitors
Humans
Malaria, Falciparum--drug therapy
Models, Molecular
Molecular Structure
Parasitic Sensitivity Tests
Plasmodium falciparum--drug effects
Saccharomyces cerevisiae--enzymology
Small Molecule Libraries--chemical synthesis
Structure-Activity Relationship