Biased Agonism and Biased Allosteric Modulation at the CB1 Cannabinoid Receptor.

Khajehali, Elham

Biased Agonism and Biased Allosteric Modulation at the CB1 Cannabinoid Receptor. [electronic resource] - Molecular pharmacology Aug 2015 - 368-79 p. digital

Publication Type: Journal Article; Research Support, Non-U.S. Gov't

1521-0111

10.1124/mol.115.099192 doi


Allosteric Regulation
Animals
Benzoxazines--pharmacology
CHO Cells
Cannabinoid Receptor Agonists--pharmacology
Cricetulus
Cyclohexanols--pharmacology
Dronabinol--analogs & derivatives
Humans
Indoles--pharmacology
MAP Kinase Signaling System--drug effects
Morpholines--pharmacology
Naphthalenes--pharmacology
Phosphorylation
Piperidines--pharmacology
Pyrazoles--pharmacology
Receptor, Cannabinoid, CB1--chemistry
Rimonabant
Signal Transduction--drug effects