Diaminothiazoles evade multidrug resistance in cancer cells and xenograft tumour models and develop transient specific resistance: understanding the basis of broad-spectrum versus specific resistance.
Vasudevan, Smreti
Diaminothiazoles evade multidrug resistance in cancer cells and xenograft tumour models and develop transient specific resistance: understanding the basis of broad-spectrum versus specific resistance. [electronic resource] - Carcinogenesis Aug 2015 - 883-93 p. digital
Publication Type: Journal Article; Research Support, Non-U.S. Gov't
1460-2180
10.1093/carcin/bgv072 doi
ATP Binding Cassette Transporter, Subfamily B--metabolism
ATP Binding Cassette Transporter, Subfamily B, Member 1--chemistry
Animals
Antineoplastic Agents--chemistry
Cell Line, Tumor--drug effects
Drug Resistance, Multiple--drug effects
Drug Resistance, Neoplasm--drug effects
Female
Humans
Male
Mice, SCID
Molecular Docking Simulation
Paclitaxel--pharmacology
Thiazoles--chemistry
Tubulin--chemistry
Xenograft Model Antitumor Assays
Diaminothiazoles evade multidrug resistance in cancer cells and xenograft tumour models and develop transient specific resistance: understanding the basis of broad-spectrum versus specific resistance. [electronic resource] - Carcinogenesis Aug 2015 - 883-93 p. digital
Publication Type: Journal Article; Research Support, Non-U.S. Gov't
1460-2180
10.1093/carcin/bgv072 doi
ATP Binding Cassette Transporter, Subfamily B--metabolism
ATP Binding Cassette Transporter, Subfamily B, Member 1--chemistry
Animals
Antineoplastic Agents--chemistry
Cell Line, Tumor--drug effects
Drug Resistance, Multiple--drug effects
Drug Resistance, Neoplasm--drug effects
Female
Humans
Male
Mice, SCID
Molecular Docking Simulation
Paclitaxel--pharmacology
Thiazoles--chemistry
Tubulin--chemistry
Xenograft Model Antitumor Assays