LP99: Discovery and Synthesis of the First Selective BRD7/9 Bromodomain Inhibitor.

Clark, Peter G K

LP99: Discovery and Synthesis of the First Selective BRD7/9 Bromodomain Inhibitor. [electronic resource] - Angewandte Chemie (International ed. in English) May 2015 - 6217-21 p. digital

Publication Type: Journal Article; Research Support, Non-U.S. Gov't

1521-3773

10.1002/anie.201501394 doi


Chromosomal Proteins, Non-Histone--antagonists & inhibitors
Drug Discovery
Humans
Lactams--chemistry
Models, Molecular
Transcription Factors--antagonists & inhibitors