Discovery of I-BRD9, a Selective Cell Active Chemical Probe for Bromodomain Containing Protein 9 Inhibition.

Theodoulou, Natalie H

Discovery of I-BRD9, a Selective Cell Active Chemical Probe for Bromodomain Containing Protein 9 Inhibition. [electronic resource] - Journal of medicinal chemistry Feb 2016 - 1425-39 p. digital

Publication Type: Journal Article; Research Support, Non-U.S. Gov't

1520-4804

10.1021/acs.jmedchem.5b00256 doi


Amino Acid Sequence
Binding Sites
Cell Line
Crystallography, X-Ray
Drug Discovery
Humans
Models, Molecular
Molecular Docking Simulation
Small Molecule Libraries--chemistry
Transcription Factors--antagonists & inhibitors