EGFR participates downstream of ERα in estradiol-17β-D-glucuronide-induced impairment of Abcc2 function in isolated rat hepatocyte couplets.
Barosso, Ismael R
EGFR participates downstream of ERα in estradiol-17β-D-glucuronide-induced impairment of Abcc2 function in isolated rat hepatocyte couplets. [electronic resource] - Archives of toxicology Apr 2016 - 891-903 p. digital
Publication Type: Journal Article; Research Support, Non-U.S. Gov't
1432-0738
10.1007/s00204-015-1507-8 doi
ATP-Binding Cassette Transporters--metabolism
Animals
Bile Canaliculi--drug effects
Cells, Cultured
Cholestasis--chemically induced
ErbB Receptors--genetics
Estradiol--analogs & derivatives
Estrogen Receptor Antagonists--pharmacology
Estrogen Receptor alpha--metabolism
Female
Fulvestrant
Gene Knockdown Techniques
Hepatocytes--drug effects
Quinazolines--pharmacology
Rats
Rats, Wistar
Tyrphostins--pharmacology
src-Family Kinases--metabolism
EGFR participates downstream of ERα in estradiol-17β-D-glucuronide-induced impairment of Abcc2 function in isolated rat hepatocyte couplets. [electronic resource] - Archives of toxicology Apr 2016 - 891-903 p. digital
Publication Type: Journal Article; Research Support, Non-U.S. Gov't
1432-0738
10.1007/s00204-015-1507-8 doi
ATP-Binding Cassette Transporters--metabolism
Animals
Bile Canaliculi--drug effects
Cells, Cultured
Cholestasis--chemically induced
ErbB Receptors--genetics
Estradiol--analogs & derivatives
Estrogen Receptor Antagonists--pharmacology
Estrogen Receptor alpha--metabolism
Female
Fulvestrant
Gene Knockdown Techniques
Hepatocytes--drug effects
Quinazolines--pharmacology
Rats
Rats, Wistar
Tyrphostins--pharmacology
src-Family Kinases--metabolism