Discovery of new thienopyrimidinone derivatives displaying antimalarial properties toward both erythrocytic and hepatic stages of Plasmodium.

Cohen, Anita

Discovery of new thienopyrimidinone derivatives displaying antimalarial properties toward both erythrocytic and hepatic stages of Plasmodium. [electronic resource] - European journal of medicinal chemistry May 2015 - 16-28 p. digital

Publication Type: Journal Article

1768-3254

10.1016/j.ejmech.2015.03.011 doi


Animals
Antimalarials--chemistry
CHO Cells
Cell Proliferation--drug effects
Cricetinae
Cricetulus
Drug Discovery
Erythrocytes--drug effects
Hep G2 Cells
Humans
Liver--drug effects
Malaria--drug therapy
Male
Mice
Parasitemia--drug therapy
Plasmodium falciparum--drug effects
Pyrimidines--chemistry
Structure-Activity Relationship
Trophozoites--drug effects