Epoxy-α-lapachone has in vitro and in vivo anti-leishmania (Leishmania) amazonensis effects and inhibits serine proteinase activity in this parasite.
Souza-Silva, Franklin
Epoxy-α-lapachone has in vitro and in vivo anti-leishmania (Leishmania) amazonensis effects and inhibits serine proteinase activity in this parasite. [electronic resource] - Antimicrobial agents and chemotherapy Apr 2015 - 1910-8 p. digital
Publication Type: Journal Article; Research Support, Non-U.S. Gov't
1098-6596
10.1128/AAC.04742-14 doi
Animals
Antipain--pharmacology
Antiprotozoal Agents--pharmacology
Computer Simulation
Leishmania mexicana--drug effects
Leishmaniasis, Cutaneous--drug therapy
Mice
Mice, Inbred BALB C
Naphthoquinones--pharmacology
Protein Binding
Serine Endopeptidases--metabolism
Serine Proteinase Inhibitors--pharmacology
Epoxy-α-lapachone has in vitro and in vivo anti-leishmania (Leishmania) amazonensis effects and inhibits serine proteinase activity in this parasite. [electronic resource] - Antimicrobial agents and chemotherapy Apr 2015 - 1910-8 p. digital
Publication Type: Journal Article; Research Support, Non-U.S. Gov't
1098-6596
10.1128/AAC.04742-14 doi
Animals
Antipain--pharmacology
Antiprotozoal Agents--pharmacology
Computer Simulation
Leishmania mexicana--drug effects
Leishmaniasis, Cutaneous--drug therapy
Mice
Mice, Inbred BALB C
Naphthoquinones--pharmacology
Protein Binding
Serine Endopeptidases--metabolism
Serine Proteinase Inhibitors--pharmacology