Tariquidar inhibits P-glycoprotein drug efflux but activates ATPase activity by blocking transition to an open conformation.
Loo, Tip W
Tariquidar inhibits P-glycoprotein drug efflux but activates ATPase activity by blocking transition to an open conformation. [electronic resource] - Biochemical pharmacology Dec 2014 - 558-66 p. digital
Publication Type: Journal Article; Research Support, Non-U.S. Gov't
1873-2968
10.1016/j.bcp.2014.10.006 doi
ATP Binding Cassette Transporter, Subfamily B, Member 1--antagonists & inhibitors
Adenosine Triphosphatases--chemistry
Animals
Cell Line
Cricetinae
Drug Resistance, Multiple
Protein Conformation
Quinolines--pharmacokinetics
Tariquidar inhibits P-glycoprotein drug efflux but activates ATPase activity by blocking transition to an open conformation. [electronic resource] - Biochemical pharmacology Dec 2014 - 558-66 p. digital
Publication Type: Journal Article; Research Support, Non-U.S. Gov't
1873-2968
10.1016/j.bcp.2014.10.006 doi
ATP Binding Cassette Transporter, Subfamily B, Member 1--antagonists & inhibitors
Adenosine Triphosphatases--chemistry
Animals
Cell Line
Cricetinae
Drug Resistance, Multiple
Protein Conformation
Quinolines--pharmacokinetics