Synthesis and biological evaluation of pyrido[2,3-d]pyrimidine-2,4-dione derivatives as eEF-2K inhibitors.

Edupuganti, Ramakrishna

Synthesis and biological evaluation of pyrido[2,3-d]pyrimidine-2,4-dione derivatives as eEF-2K inhibitors. [electronic resource] - Bioorganic & medicinal chemistry Sep 2014 - 4910-6 p. digital

Publication Type: Journal Article; Research Support, N.I.H., Extramural

1464-3391

10.1016/j.bmc.2014.06.050 doi


Dose-Response Relationship, Drug
Elongation Factor 2 Kinase--antagonists & inhibitors
Humans
Molecular Structure
Protein Kinase Inhibitors--chemical synthesis
Pyridines--chemical synthesis
Pyrimidinones--chemical synthesis
Recombinant Proteins--metabolism
Structure-Activity Relationship
Tumor Cells, Cultured