High throughput screen identifies small molecule inhibitors specific for Mycobacterium tuberculosis phosphoserine phosphatase.
Arora, Garima
High throughput screen identifies small molecule inhibitors specific for Mycobacterium tuberculosis phosphoserine phosphatase. [electronic resource] - The Journal of biological chemistry Sep 2014 - 25149-65 p. digital
Publication Type: Journal Article; Research Support, Non-U.S. Gov't
1083-351X
10.1074/jbc.M114.597682 doi
Amino Acid Sequence
Antitubercular Agents--chemistry
Bacterial Proteins--chemistry
Cell Line, Tumor
Enzyme Inhibitors--chemistry
High-Throughput Screening Assays--methods
Humans
Kinetics
Microbial Sensitivity Tests
Models, Molecular
Molecular Sequence Data
Molecular Structure
Mycobacterium tuberculosis--drug effects
Novobiocin--analogs & derivatives
Phosphoric Monoester Hydrolases--antagonists & inhibitors
Phylogeny
Protein Binding
Protein Structure, Tertiary
Rosaniline Dyes--chemistry
Sequence Homology, Amino Acid
Small Molecule Libraries--chemistry
High throughput screen identifies small molecule inhibitors specific for Mycobacterium tuberculosis phosphoserine phosphatase. [electronic resource] - The Journal of biological chemistry Sep 2014 - 25149-65 p. digital
Publication Type: Journal Article; Research Support, Non-U.S. Gov't
1083-351X
10.1074/jbc.M114.597682 doi
Amino Acid Sequence
Antitubercular Agents--chemistry
Bacterial Proteins--chemistry
Cell Line, Tumor
Enzyme Inhibitors--chemistry
High-Throughput Screening Assays--methods
Humans
Kinetics
Microbial Sensitivity Tests
Models, Molecular
Molecular Sequence Data
Molecular Structure
Mycobacterium tuberculosis--drug effects
Novobiocin--analogs & derivatives
Phosphoric Monoester Hydrolases--antagonists & inhibitors
Phylogeny
Protein Binding
Protein Structure, Tertiary
Rosaniline Dyes--chemistry
Sequence Homology, Amino Acid
Small Molecule Libraries--chemistry