Discovery of Q203, a potent clinical candidate for the treatment of tuberculosis.

Pethe, Kevin

Discovery of Q203, a potent clinical candidate for the treatment of tuberculosis. [electronic resource] - Nature medicine Sep 2013 - 1157-60 p. digital

Publication Type: Journal Article; Research Support, Non-U.S. Gov't

1546-170X

10.1038/nm.3262 doi


Adenosine Triphosphate--biosynthesis
Animals
Cell Proliferation--drug effects
Disease Models, Animal
Drug Evaluation, Preclinical
Electron Transport Complex III--antagonists & inhibitors
Extensively Drug-Resistant Tuberculosis--drug therapy
Imidazoles--pharmacokinetics
Mice
Mice, Inbred BALB C
Mycobacterium tuberculosis--drug effects
Piperidines--pharmacokinetics
Pyridines--pharmacokinetics
Rats
Rats, Sprague-Dawley