Discovery of a novel series of quinolone α7 nicotinic acetylcholine receptor agonists.

McDonald, Ivar M

Discovery of a novel series of quinolone α7 nicotinic acetylcholine receptor agonists. [electronic resource] - Bioorganic & medicinal chemistry letters Mar 2013 - 1684-8 p. digital

Publication Type: Journal Article

1464-3405

10.1016/j.bmcl.2013.01.070 doi


Animals
Caco-2 Cells
Drug Evaluation, Preclinical
Humans
Kinetics
Nicotinic Agonists--chemical synthesis
Quinolones--chemical synthesis
Rats
Receptors, Nicotinic--chemistry
Structure-Activity Relationship
alpha7 Nicotinic Acetylcholine Receptor