In vivo and ex vivo inhibition of spinal nerve ligation-induced ectopic activity by sodium channel blockers correlate to in vitro inhibition of NaV1.7 and clinical efficacy: a pharmacokinetic-pharmacodynamic translational approach.
Kalezic, Ivana
In vivo and ex vivo inhibition of spinal nerve ligation-induced ectopic activity by sodium channel blockers correlate to in vitro inhibition of NaV1.7 and clinical efficacy: a pharmacokinetic-pharmacodynamic translational approach. [electronic resource] - Pharmaceutical research May 2013 - 1409-22 p. digital
Publication Type: Journal Article
1573-904X
10.1007/s11095-013-0979-6 doi
Animals
HEK293 Cells
Humans
Ligation
Male
NAV1.7 Voltage-Gated Sodium Channel--metabolism
Neuralgia--drug therapy
Rats
Rats, Sprague-Dawley
Sodium Channel Blockers--blood
Spinal Nerves--drug effects
In vivo and ex vivo inhibition of spinal nerve ligation-induced ectopic activity by sodium channel blockers correlate to in vitro inhibition of NaV1.7 and clinical efficacy: a pharmacokinetic-pharmacodynamic translational approach. [electronic resource] - Pharmaceutical research May 2013 - 1409-22 p. digital
Publication Type: Journal Article
1573-904X
10.1007/s11095-013-0979-6 doi
Animals
HEK293 Cells
Humans
Ligation
Male
NAV1.7 Voltage-Gated Sodium Channel--metabolism
Neuralgia--drug therapy
Rats
Rats, Sprague-Dawley
Sodium Channel Blockers--blood
Spinal Nerves--drug effects