Distinct CCK-2 receptor conformations associated with β-arrestin-2 recruitment or phospholipase-C activation revealed by a biased antagonist.
Magnan, Rémi
Distinct CCK-2 receptor conformations associated with β-arrestin-2 recruitment or phospholipase-C activation revealed by a biased antagonist. [electronic resource] - Journal of the American Chemical Society Feb 2013 - 2560-73 p. digital
Publication Type: Journal Article; Research Support, Non-U.S. Gov't
1520-5126
10.1021/ja308784w doi
Adamantane--analogs & derivatives
Arrestins--chemistry
Binding Sites
Enzyme Activation--drug effects
Humans
Microscopy, Confocal
Models, Molecular
Molecular Structure
Mutation
Phenylurea Compounds--pharmacology
Protein Conformation
Receptor, Cholecystokinin B--antagonists & inhibitors
Signal Transduction
Type C Phospholipases--chemistry
Up-Regulation
beta-Arrestin 2
beta-Arrestins
Distinct CCK-2 receptor conformations associated with β-arrestin-2 recruitment or phospholipase-C activation revealed by a biased antagonist. [electronic resource] - Journal of the American Chemical Society Feb 2013 - 2560-73 p. digital
Publication Type: Journal Article; Research Support, Non-U.S. Gov't
1520-5126
10.1021/ja308784w doi
Adamantane--analogs & derivatives
Arrestins--chemistry
Binding Sites
Enzyme Activation--drug effects
Humans
Microscopy, Confocal
Models, Molecular
Molecular Structure
Mutation
Phenylurea Compounds--pharmacology
Protein Conformation
Receptor, Cholecystokinin B--antagonists & inhibitors
Signal Transduction
Type C Phospholipases--chemistry
Up-Regulation
beta-Arrestin 2
beta-Arrestins