The precise chemical-physical nature of the pharmacore in FK506 binding protein inhibition: ElteX, a New class of nanomolar FKBP12 ligands.

Martina, Maria Raffaella

The precise chemical-physical nature of the pharmacore in FK506 binding protein inhibition: ElteX, a New class of nanomolar FKBP12 ligands. [electronic resource] - Journal of medicinal chemistry Feb 2013 - 1041-51 p. digital

Publication Type: Journal Article; Research Support, Non-U.S. Gov't

1520-4804

10.1021/jm3015052 doi


Fluorescence
Ligands
Models, Molecular
Piperidines--chemistry
Protein Binding
Tacrolimus--metabolism
Tacrolimus Binding Protein 1A--metabolism