Heteroaryl urea inhibitors of fatty acid amide hydrolase: structure-mutagenicity relationships for arylamine metabolites.
Tichenor, Mark S
Heteroaryl urea inhibitors of fatty acid amide hydrolase: structure-mutagenicity relationships for arylamine metabolites. [electronic resource] - Bioorganic & medicinal chemistry letters Dec 2012 - 7357-62 p. digital
Publication Type: Journal Article
1464-3405
10.1016/j.bmcl.2012.10.076 doi
Amidohydrolases--antagonists & inhibitors
Amines--metabolism
Animals
Dose-Response Relationship, Drug
Enzyme Inhibitors--chemical synthesis
Humans
Mixed Function Oxygenases--metabolism
Molecular Structure
Mutagenicity Tests
Mutagens--metabolism
Rats
Structure-Activity Relationship
Urea--analogs & derivatives
Heteroaryl urea inhibitors of fatty acid amide hydrolase: structure-mutagenicity relationships for arylamine metabolites. [electronic resource] - Bioorganic & medicinal chemistry letters Dec 2012 - 7357-62 p. digital
Publication Type: Journal Article
1464-3405
10.1016/j.bmcl.2012.10.076 doi
Amidohydrolases--antagonists & inhibitors
Amines--metabolism
Animals
Dose-Response Relationship, Drug
Enzyme Inhibitors--chemical synthesis
Humans
Mixed Function Oxygenases--metabolism
Molecular Structure
Mutagenicity Tests
Mutagens--metabolism
Rats
Structure-Activity Relationship
Urea--analogs & derivatives