Characterisation of the roles of ABCB1, ABCC1, ABCC2 and ABCG2 in the transport and pharmacokinetics of actinomycin D in vitro and in vivo.
Hill, Christopher R
Characterisation of the roles of ABCB1, ABCC1, ABCC2 and ABCG2 in the transport and pharmacokinetics of actinomycin D in vitro and in vivo. [electronic resource] - Biochemical pharmacology Jan 2013 - 29-37 p. digital
Publication Type: Journal Article; Research Support, Non-U.S. Gov't
1873-2968
10.1016/j.bcp.2012.10.004 doi
ATP Binding Cassette Transporter, Subfamily B
ATP Binding Cassette Transporter, Subfamily B, Member 1--genetics
ATP Binding Cassette Transporter, Subfamily G, Member 2
ATP-Binding Cassette Transporters--metabolism
Animals
Antibiotics, Antineoplastic--blood
Biological Transport
Cell Proliferation--drug effects
Dactinomycin--blood
Dogs
Doxorubicin--pharmacokinetics
Humans
Madin Darby Canine Kidney Cells
Mice
Mice, Knockout
Multidrug Resistance-Associated Protein 2
Multidrug Resistance-Associated Proteins--genetics
Neoplasm Proteins--metabolism
Tissue Distribution
Characterisation of the roles of ABCB1, ABCC1, ABCC2 and ABCG2 in the transport and pharmacokinetics of actinomycin D in vitro and in vivo. [electronic resource] - Biochemical pharmacology Jan 2013 - 29-37 p. digital
Publication Type: Journal Article; Research Support, Non-U.S. Gov't
1873-2968
10.1016/j.bcp.2012.10.004 doi
ATP Binding Cassette Transporter, Subfamily B
ATP Binding Cassette Transporter, Subfamily B, Member 1--genetics
ATP Binding Cassette Transporter, Subfamily G, Member 2
ATP-Binding Cassette Transporters--metabolism
Animals
Antibiotics, Antineoplastic--blood
Biological Transport
Cell Proliferation--drug effects
Dactinomycin--blood
Dogs
Doxorubicin--pharmacokinetics
Humans
Madin Darby Canine Kidney Cells
Mice
Mice, Knockout
Multidrug Resistance-Associated Protein 2
Multidrug Resistance-Associated Proteins--genetics
Neoplasm Proteins--metabolism
Tissue Distribution