Blockade of STAT3 activation by sorafenib derivatives through enhancing SHP-1 phosphatase activity.
Chen, Kuen-Feng
Blockade of STAT3 activation by sorafenib derivatives through enhancing SHP-1 phosphatase activity. [electronic resource] - European journal of medicinal chemistry Sep 2012 - 220-7 p. digital
Publication Type: Journal Article; Research Support, Non-U.S. Gov't
1768-3254
10.1016/j.ejmech.2012.07.023 doi
Animals
Benzenesulfonates--chemistry
Cell Line, Tumor
Dose-Response Relationship, Drug
Down-Regulation--drug effects
Humans
Male
Mice
Mice, Nude
Niacinamide--analogs & derivatives
Phenylurea Compounds
Phosphoproteins--metabolism
Protein Kinase Inhibitors--analogs & derivatives
Protein Kinases--metabolism
Protein Tyrosine Phosphatase, Non-Receptor Type 6--metabolism
Pyridines--chemistry
STAT3 Transcription Factor--metabolism
Sorafenib
Xenograft Model Antitumor Assays
Blockade of STAT3 activation by sorafenib derivatives through enhancing SHP-1 phosphatase activity. [electronic resource] - European journal of medicinal chemistry Sep 2012 - 220-7 p. digital
Publication Type: Journal Article; Research Support, Non-U.S. Gov't
1768-3254
10.1016/j.ejmech.2012.07.023 doi
Animals
Benzenesulfonates--chemistry
Cell Line, Tumor
Dose-Response Relationship, Drug
Down-Regulation--drug effects
Humans
Male
Mice
Mice, Nude
Niacinamide--analogs & derivatives
Phenylurea Compounds
Phosphoproteins--metabolism
Protein Kinase Inhibitors--analogs & derivatives
Protein Kinases--metabolism
Protein Tyrosine Phosphatase, Non-Receptor Type 6--metabolism
Pyridines--chemistry
STAT3 Transcription Factor--metabolism
Sorafenib
Xenograft Model Antitumor Assays