Development of isoform selective PI3-kinase inhibitors as pharmacological tools for elucidating the PI3K pathway.
Bruce, Ian
Development of isoform selective PI3-kinase inhibitors as pharmacological tools for elucidating the PI3K pathway. [electronic resource] - Bioorganic & medicinal chemistry letters Sep 2012 - 5445-50 p. digital
Publication Type: Journal Article
1464-3405
10.1016/j.bmcl.2012.07.042 doi
Animals
Catalytic Domain
Female
Humans
Mice
Models, Molecular
Phosphatidylinositol 3-Kinases--chemistry
Phosphoinositide-3 Kinase Inhibitors
Protein Isoforms--antagonists & inhibitors
Protein Kinase Inhibitors--chemistry
Rats
Signal Transduction--drug effects
Thiazoles--chemistry
Development of isoform selective PI3-kinase inhibitors as pharmacological tools for elucidating the PI3K pathway. [electronic resource] - Bioorganic & medicinal chemistry letters Sep 2012 - 5445-50 p. digital
Publication Type: Journal Article
1464-3405
10.1016/j.bmcl.2012.07.042 doi
Animals
Catalytic Domain
Female
Humans
Mice
Models, Molecular
Phosphatidylinositol 3-Kinases--chemistry
Phosphoinositide-3 Kinase Inhibitors
Protein Isoforms--antagonists & inhibitors
Protein Kinase Inhibitors--chemistry
Rats
Signal Transduction--drug effects
Thiazoles--chemistry