A combined targeted/phenotypic approach for the identification of new antiangiogenics agents active on a zebrafish model: from in silico screening to cyclodextrin formulation.
Radi, Marco
A combined targeted/phenotypic approach for the identification of new antiangiogenics agents active on a zebrafish model: from in silico screening to cyclodextrin formulation. [electronic resource] - Bioorganic & medicinal chemistry letters Sep 2012 - 5579-83 p. digital
Publication Type: Journal Article; Research Support, Non-U.S. Gov't
1464-3405
10.1016/j.bmcl.2012.07.014 doi
Angiogenesis Inhibitors--chemistry
Animals
Cyclodextrins--chemistry
Drug Carriers--chemistry
Drug Discovery--methods
Embryo, Nonmammalian--blood supply
Human Umbilical Vein Endothelial Cells
Humans
Models, Animal
Neovascularization, Pathologic--drug therapy
Neovascularization, Physiologic--drug effects
Proto-Oncogene Proteins pp60(c-src)--antagonists & inhibitors
Vascular Endothelial Growth Factor Receptor-2--antagonists & inhibitors
Zebrafish--embryology
A combined targeted/phenotypic approach for the identification of new antiangiogenics agents active on a zebrafish model: from in silico screening to cyclodextrin formulation. [electronic resource] - Bioorganic & medicinal chemistry letters Sep 2012 - 5579-83 p. digital
Publication Type: Journal Article; Research Support, Non-U.S. Gov't
1464-3405
10.1016/j.bmcl.2012.07.014 doi
Angiogenesis Inhibitors--chemistry
Animals
Cyclodextrins--chemistry
Drug Carriers--chemistry
Drug Discovery--methods
Embryo, Nonmammalian--blood supply
Human Umbilical Vein Endothelial Cells
Humans
Models, Animal
Neovascularization, Pathologic--drug therapy
Neovascularization, Physiologic--drug effects
Proto-Oncogene Proteins pp60(c-src)--antagonists & inhibitors
Vascular Endothelial Growth Factor Receptor-2--antagonists & inhibitors
Zebrafish--embryology