Evaluation of potential Myt1 kinase inhibitors by TR-FRET based binding assay.
Rohe, Alexander
Evaluation of potential Myt1 kinase inhibitors by TR-FRET based binding assay. [electronic resource] - European journal of medicinal chemistry Mar 2013 - 41-8 p. digital
Publication Type: Journal Article; Research Support, Non-U.S. Gov't
1768-3254
10.1016/j.ejmech.2012.06.007 doi
Dose-Response Relationship, Drug
Fluorescence Resonance Energy Transfer
Glycolipids--chemical synthesis
Humans
Membrane Proteins--antagonists & inhibitors
Models, Molecular
Molecular Structure
Protein Kinase Inhibitors--chemical synthesis
Protein Serine-Threonine Kinases--antagonists & inhibitors
Protein-Tyrosine Kinases--antagonists & inhibitors
Structure-Activity Relationship
Evaluation of potential Myt1 kinase inhibitors by TR-FRET based binding assay. [electronic resource] - European journal of medicinal chemistry Mar 2013 - 41-8 p. digital
Publication Type: Journal Article; Research Support, Non-U.S. Gov't
1768-3254
10.1016/j.ejmech.2012.06.007 doi
Dose-Response Relationship, Drug
Fluorescence Resonance Energy Transfer
Glycolipids--chemical synthesis
Humans
Membrane Proteins--antagonists & inhibitors
Models, Molecular
Molecular Structure
Protein Kinase Inhibitors--chemical synthesis
Protein Serine-Threonine Kinases--antagonists & inhibitors
Protein-Tyrosine Kinases--antagonists & inhibitors
Structure-Activity Relationship