Synthesis and structure-activity relationships of pyrido[3,2-b]pyrazin-3(4H)-ones and pteridin-7(8H)-ones as corticotropin-releasing factor-1 receptor antagonists.
Dzierba, Carolyn D
Synthesis and structure-activity relationships of pyrido[3,2-b]pyrazin-3(4H)-ones and pteridin-7(8H)-ones as corticotropin-releasing factor-1 receptor antagonists. [electronic resource] - Bioorganic & medicinal chemistry letters Aug 2012 - 4986-9 p. digital
Publication Type: Journal Article
1464-3405
10.1016/j.bmcl.2012.06.034 doi
Animals
Anti-Anxiety Agents--chemical synthesis
Half-Life
Pteridines--chemical synthesis
Pyrazines--chemical synthesis
Rats
Receptors, Corticotropin-Releasing Hormone--antagonists & inhibitors
Structure-Activity Relationship
CRF Receptor, Type 1
Synthesis and structure-activity relationships of pyrido[3,2-b]pyrazin-3(4H)-ones and pteridin-7(8H)-ones as corticotropin-releasing factor-1 receptor antagonists. [electronic resource] - Bioorganic & medicinal chemistry letters Aug 2012 - 4986-9 p. digital
Publication Type: Journal Article
1464-3405
10.1016/j.bmcl.2012.06.034 doi
Animals
Anti-Anxiety Agents--chemical synthesis
Half-Life
Pteridines--chemical synthesis
Pyrazines--chemical synthesis
Rats
Receptors, Corticotropin-Releasing Hormone--antagonists & inhibitors
Structure-Activity Relationship
CRF Receptor, Type 1