Phase I pharmacologic and pharmacodynamic study of the gamma secretase (Notch) inhibitor MK-0752 in adult patients with advanced solid tumors.
Krop, Ian
Phase I pharmacologic and pharmacodynamic study of the gamma secretase (Notch) inhibitor MK-0752 in adult patients with advanced solid tumors. [electronic resource] - Journal of clinical oncology : official journal of the American Society of Clinical Oncology Jul 2012 - 2307-13 p. digital
Publication Type: Clinical Trial, Phase I; Journal Article; Multicenter Study; Research Support, Non-U.S. Gov't
1527-7755
10.1200/JCO.2011.39.1540 doi
Administration, Oral
Adult
Aged
Aged, 80 and over
Amyloid Precursor Protein Secretases--antagonists & inhibitors
Benzene Derivatives
Cohort Studies
Dose-Response Relationship, Drug
Drug Administration Schedule
Female
Humans
Male
Middle Aged
Neoplasms--drug therapy
Propionates--adverse effects
Sulfones--adverse effects
Treatment Outcome
Phase I pharmacologic and pharmacodynamic study of the gamma secretase (Notch) inhibitor MK-0752 in adult patients with advanced solid tumors. [electronic resource] - Journal of clinical oncology : official journal of the American Society of Clinical Oncology Jul 2012 - 2307-13 p. digital
Publication Type: Clinical Trial, Phase I; Journal Article; Multicenter Study; Research Support, Non-U.S. Gov't
1527-7755
10.1200/JCO.2011.39.1540 doi
Administration, Oral
Adult
Aged
Aged, 80 and over
Amyloid Precursor Protein Secretases--antagonists & inhibitors
Benzene Derivatives
Cohort Studies
Dose-Response Relationship, Drug
Drug Administration Schedule
Female
Humans
Male
Middle Aged
Neoplasms--drug therapy
Propionates--adverse effects
Sulfones--adverse effects
Treatment Outcome