Identification of ETP-46321, a potent and orally bioavailable PI3K α, δ inhibitor.
Martínez González, Sonia
Identification of ETP-46321, a potent and orally bioavailable PI3K α, δ inhibitor. [electronic resource] - Bioorganic & medicinal chemistry letters May 2012 - 3460-6 p. digital
Publication Type: Journal Article; Research Support, Non-U.S. Gov't
1464-3405
10.1016/j.bmcl.2012.03.090 doi
Administration, Oral
Biological Availability
Humans
Imidazoles--administration & dosage
Isoenzymes--antagonists & inhibitors
Phosphoinositide-3 Kinase Inhibitors
Positron-Emission Tomography
Protein Kinase Inhibitors--administration & dosage
Pyrazines--administration & dosage
Tomography, X-Ray Computed
Identification of ETP-46321, a potent and orally bioavailable PI3K α, δ inhibitor. [electronic resource] - Bioorganic & medicinal chemistry letters May 2012 - 3460-6 p. digital
Publication Type: Journal Article; Research Support, Non-U.S. Gov't
1464-3405
10.1016/j.bmcl.2012.03.090 doi
Administration, Oral
Biological Availability
Humans
Imidazoles--administration & dosage
Isoenzymes--antagonists & inhibitors
Phosphoinositide-3 Kinase Inhibitors
Positron-Emission Tomography
Protein Kinase Inhibitors--administration & dosage
Pyrazines--administration & dosage
Tomography, X-Ray Computed