Identification of ETP-46321, a potent and orally bioavailable PI3K α, δ inhibitor.

Martínez González, Sonia

Identification of ETP-46321, a potent and orally bioavailable PI3K α, δ inhibitor. [electronic resource] - Bioorganic & medicinal chemistry letters May 2012 - 3460-6 p. digital

Publication Type: Journal Article; Research Support, Non-U.S. Gov't

1464-3405

10.1016/j.bmcl.2012.03.090 doi


Administration, Oral
Biological Availability
Humans
Imidazoles--administration & dosage
Isoenzymes--antagonists & inhibitors
Phosphoinositide-3 Kinase Inhibitors
Positron-Emission Tomography
Protein Kinase Inhibitors--administration & dosage
Pyrazines--administration & dosage
Tomography, X-Ray Computed