Stress is a critical player in CYP3A, CYP2C, and CYP2D regulation: role of adrenergic receptor signaling pathways.
Daskalopoulos, Evangelos P
Stress is a critical player in CYP3A, CYP2C, and CYP2D regulation: role of adrenergic receptor signaling pathways. [electronic resource] - American journal of physiology. Endocrinology and metabolism Jul 2012 - E40-54 p. digital
Publication Type: Journal Article
1522-1555
10.1152/ajpendo.00545.2011 doi
Adrenergic Agonists--pharmacology
Animals
Aryl Hydrocarbon Hydroxylases--genetics
Cells, Cultured
Corticosterone--metabolism
Cytochrome P-450 CYP2D6--genetics
Cytochrome P-450 CYP3A--genetics
Cytochrome P450 Family 2
Enzyme Induction--drug effects
Epinephrine--metabolism
Hepatocytes--cytology
Isoenzymes--genetics
Male
Maternal Deprivation
Protein Kinase Inhibitors--pharmacology
RNA, Messenger--metabolism
Rats
Rats, Wistar
Receptors, Adrenergic--chemistry
Restraint, Physical--adverse effects
Signal Transduction--drug effects
Steroid 16-alpha-Hydroxylase--genetics
Stress, Physiological
Stress, Psychological--metabolism
Stress is a critical player in CYP3A, CYP2C, and CYP2D regulation: role of adrenergic receptor signaling pathways. [electronic resource] - American journal of physiology. Endocrinology and metabolism Jul 2012 - E40-54 p. digital
Publication Type: Journal Article
1522-1555
10.1152/ajpendo.00545.2011 doi
Adrenergic Agonists--pharmacology
Animals
Aryl Hydrocarbon Hydroxylases--genetics
Cells, Cultured
Corticosterone--metabolism
Cytochrome P-450 CYP2D6--genetics
Cytochrome P-450 CYP3A--genetics
Cytochrome P450 Family 2
Enzyme Induction--drug effects
Epinephrine--metabolism
Hepatocytes--cytology
Isoenzymes--genetics
Male
Maternal Deprivation
Protein Kinase Inhibitors--pharmacology
RNA, Messenger--metabolism
Rats
Rats, Wistar
Receptors, Adrenergic--chemistry
Restraint, Physical--adverse effects
Signal Transduction--drug effects
Steroid 16-alpha-Hydroxylase--genetics
Stress, Physiological
Stress, Psychological--metabolism