Impact of CYP3A5 and ABCB1 gene polymorphisms on fentanyl pharmacokinetics and clinical responses in cancer patients undergoing conversion to a transdermal system.
Takashina, Yoshiaki
Impact of CYP3A5 and ABCB1 gene polymorphisms on fentanyl pharmacokinetics and clinical responses in cancer patients undergoing conversion to a transdermal system. [electronic resource] - Drug metabolism and pharmacokinetics 2012 - 414-21 p. digital
Publication Type: Journal Article; Research Support, Non-U.S. Gov't
1880-0920
10.2133/dmpk.dmpk-11-rg-134 doi
ATP Binding Cassette Transporter, Subfamily B
ATP Binding Cassette Transporter, Subfamily B, Member 1--genetics
Administration, Cutaneous
Aged
Analgesics, Opioid--administration & dosage
Cytochrome P-450 CYP3A--genetics
Drug Monitoring
Female
Fentanyl--administration & dosage
Genotype
Humans
Japan
Logistic Models
Male
Middle Aged
Neoplasms--drug therapy
Odds Ratio
Pharmacogenetics
Phenotype
Polymorphism, Genetic
Impact of CYP3A5 and ABCB1 gene polymorphisms on fentanyl pharmacokinetics and clinical responses in cancer patients undergoing conversion to a transdermal system. [electronic resource] - Drug metabolism and pharmacokinetics 2012 - 414-21 p. digital
Publication Type: Journal Article; Research Support, Non-U.S. Gov't
1880-0920
10.2133/dmpk.dmpk-11-rg-134 doi
ATP Binding Cassette Transporter, Subfamily B
ATP Binding Cassette Transporter, Subfamily B, Member 1--genetics
Administration, Cutaneous
Aged
Analgesics, Opioid--administration & dosage
Cytochrome P-450 CYP3A--genetics
Drug Monitoring
Female
Fentanyl--administration & dosage
Genotype
Humans
Japan
Logistic Models
Male
Middle Aged
Neoplasms--drug therapy
Odds Ratio
Pharmacogenetics
Phenotype
Polymorphism, Genetic