Discovery of a new class of potent prolylcarboxypeptidase inhibitors derived from alanine.

Wu, Zhicai

Discovery of a new class of potent prolylcarboxypeptidase inhibitors derived from alanine. [electronic resource] - Bioorganic & medicinal chemistry letters Feb 2012 - 1774-8 p. digital

Publication Type: Journal Article

1464-3405

10.1016/j.bmcl.2011.12.064 doi


Alanine--chemistry
Animals
Carboxypeptidases--antagonists & inhibitors
Drug Discovery
Enzyme Activation--drug effects
Enzyme Inhibitors--chemical synthesis
Humans
Inhibitory Concentration 50
Mice
Molecular Structure
Structure-Activity Relationship