Involvement of concentrative nucleoside transporter 1 in intestinal absorption of trifluorothymidine, a novel antitumor nucleoside, in rats.

Okayama, Takashige

Involvement of concentrative nucleoside transporter 1 in intestinal absorption of trifluorothymidine, a novel antitumor nucleoside, in rats. [electronic resource] - The Journal of pharmacology and experimental therapeutics Feb 2012 - 457-62 p. digital

Publication Type: Journal Article

1521-0103

10.1124/jpet.111.186296 doi


2,4-Dinitrophenol--pharmacology
Animals
Antineoplastic Agents--administration & dosage
Binding, Competitive--physiology
Drug Interactions--physiology
Female
Inosine--metabolism
Intestinal Absorption--drug effects
Intestinal Mucosa--chemistry
Jejunum--drug effects
Kinetics
Male
Membrane Transport Proteins--genetics
Oocytes--metabolism
Perfusion--methods
RNA--administration & dosage
RNA, Complementary--administration & dosage
Rats
Rats, Sprague-Dawley
Sodium Azide--pharmacology
Thymidine--analogs & derivatives
Thymidine Phosphorylase--antagonists & inhibitors
Thymidylate Synthase--antagonists & inhibitors
Trifluridine--administration & dosage
Uridine--pharmacology
Xenopus laevis